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GPCR/G protein

G protein–coupled receptors (GPCRs) which are also known as seven-transmembrane domain receptors, 7TM receptors, heptahelical receptors, serpentine receptor, and G protein–linked receptors (GPLR), constitute a large protein family of receptors, that detect molecules outside the cell and activate internal signal transduction pathways and, ultimately, cellular responses. Coupling with G proteins, they are called seven-transmembrane receptors because they pass through the cell membrane seven times.

Products for GPCR/G protein

  1. Cat.No. Product Name Information
  2. BCN2191 Adrenaline Adrenaline
  3. BCN2203 Corticosterone Endogenous glucocorticoid Corticosterone
  4. BCN2167 Fingolimod hydrochloride Fingolimod hydrochloride
  5. BCN4344 Grifolic acid Selective partial FFA4 (GPR120) agonist Grifolic acid
  6. BCN2192 Hydrocortisone Adrenal glucocorticoid; immunosuppressant Hydrocortisone
  7. BCN4128 Phloretin Phloretin
  8. BCN1940 Scopine Scopine
  9. BCN2164 Silodosin Silodosin
  10. BCC1082 CP-945598 HCl CB1 receptor antagonist CP-945598 HCl
  11. BCC1102 GW9508 Potent and selective FFA1 (GPR40) agonist GW9508
  12. BCC1107 Ramelteon Agonist of melatonin receptor(M1-M2),highly selective Ramelteon
  13. BCC1142 Macitentan Endothelin (ET)(A) and ET(B) receptor antagonist Macitentan
  14. BCC1155 Ki16425 LPA1 and LPA3 receptor antagonist Ki16425
  15. BCC1158 Plerixafor (AMD3100) CXCR4 chemokine receptor antagonist Plerixafor (AMD3100)
  16. BCC1257 Doxazosin Mesylate α1-adrenergic receptor antagonist Doxazosin Mesylate
  17. BCC1293 (R,R)-Formoterol β2-selective adrenergic agonist (R,R)-Formoterol
  18. BCC1312 5-Iodotubercidin Potent adenosine kinase inhibitor; decreases DNA methylation 5-Iodotubercidin
  19. BCC1332 AH 6809 EP1 and EP2 receptor antagonist AH 6809
  20. BCC1351 AM095 Potent LPA1 receptor antagonist AM095
  21. BCC1352 AM-095 free base Potent LPA1 receptor antagonist AM-095 free base
  22. BCC1353 AM630 CB2 selective antagonist/inverse agonist AM630
  23. BCC1355 AM966 LPA1 antagonist, oral active, high affinity, selective, AM966
  24. BCC1357 AMD-070 CXCR4 antagonist,potent and selective AMD-070
  25. BCC1358 AMD-070 hydrochloride CXCR4 antagonist,potent and selective AMD-070 hydrochloride
  26. BCC1362 Anamorelin Ghrelin receptor agonist, synthetic, orally active Anamorelin
  27. BCC1363 Anamorelin Fumarate GHSR stimulator Anamorelin Fumarate
  28. BCC1364 Anamorelin hydrochloride GHSR/ghrelin receptor agonist Anamorelin hydrochloride
  29. BCC1379 Atrasentan Endothelin antagonist receptor Atrasentan
  30. BCC1380 Atrasentan hydrochloride Endothelin antagonist receptor Atrasentan hydrochloride
  31. BCC1387 Avosentan ETA receptor antagonist Avosentan
  32. BCC1398 BAN ORL 24 NOP receptor antagonist, potent and selective BAN ORL 24
  33. BCC1448 Calcium-Sensing Receptor Antagonists I CaSR antagonist Calcium-Sensing Receptor Antagonists I
  34. BCC1450 Capadenoson Adenosine A1 receptor agonist Capadenoson
  35. BCC1460 CCG-63802 Inhibitor of regulator of G-protein signaling 4 (RGS4) protein CCG-63802
  36. BCC1461 CCG-63808 Reversible RGS inhibitor CCG-63808
  37. BCC1475 CGS 21680 Adenosine A2 receptor agonists,potent and selective CGS 21680
  38. BCC1483 Cinacalcet Cinacalcet
  39. BCC1501 CPPHA MGluR5 receptor allosteric modulator CPPHA
  40. BCC1525 Desmopressin Synthetic vasopressin analog; V1B and V2 agonist Desmopressin
  41. BCC1526 Desmopressin Acetate Synthetic analogue of arginine vasopressin Desmopressin Acetate
  42. BCC1531 Dipraglurant Dipraglurant
  43. BCC1539 DY131 ERRγ agonist DY131
  44. BCC1568 Exendin-4 Potent GLP-1 receptor agonist Exendin-4
  45. BCC1593 glucagon receptor antagonists 1 Glucagon receptor antagonist,highly potent glucagon receptor antagonists 1
  46. BCC1594 glucagon receptor antagonists 2 Glucagon receptor antagonist,highly potent glucagon receptor antagonists 2
  47. BCC1595 glucagon receptor antagonists 3 glucagon receptor antagonists 3
  48. BCC1596 Glucocorticoid receptor agonist Glucocorticoid receptor agonist
  49. BCC1599 GPR120 modulator 1 GPR120 modulator GPR120 modulator 1
  50. BCC1600 GPR120 modulator 2 GPR120 modulator GPR120 modulator 2
  51. BCC1609 Guanfacine hydrochloride α2A-adrenoceptor agonist Guanfacine hydrochloride
  52. BCC1610 GW-1100 GPR40 antagonist GW-1100
  53. BCC1634 HOKU-81 Bronchodilators,metabolite of tulobuterol HOKU-81
  54. BCC1638 Ibutamoren Mesylate High affinity ghrelin receptor agonist Ibutamoren Mesylate
  55. BCC1646 INCB 3284 dimesylate Selective CCR2 antagonist INCB 3284 dimesylate
  56. BCC1648 INCB3344 CCR2 chemokine receptor antagonist INCB3344
  57. BCC1649 INCB8761(PF-4136309) INCB8761(PF-4136309)
  58. BCC1650 Indacaterol β2-agonist Indacaterol
  59. BCC1674 JWH 073 CB1 receptor agonist JWH 073
  60. BCC1688 Laropiprant DP1 receptor antagonist,potent and selective Laropiprant
  61. BCC1710 LUF6000 A3 AR modulator LUF6000
  62. BCC1724 LY341495 Group II/III antagonist LY341495
  63. BCC1732 MBX-2982 GPR119 agonist,selective and orally-available MBX-2982
  64. BCC1736 Medetomidine α2-adrenoceptor agonist Medetomidine
  65. BCC1745 mGlu2 agonist Anti-depressants,novel potent agent mGlu2 agonist
  66. BCC1752 MK 0893 Glucagon receptor/IGF-1R antagonist MK 0893
  67. BCC1755 MK-0812 antagonist of chemokine receptor CCR-2 MK-0812
  68. BCC1757 MK-2894 EP4 receptor inhibitor MK-2894
  69. BCC1758 MK-2894 sodium salt EP4 antagonist MK-2894 sodium salt
  70. BCC1760 MK-4305 OX1/OX2 atagonist,potent and selective MK-4305
  71. BCC1767 MK-6892 Highly potential GPR109A agonist MK-6892
  72. BCC1777 MPEP Hydrochloride Positive allosteric modulator at mGlu4 and mGlu5 antagonist MPEP Hydrochloride
  73. BCC1780 MTEP hydrochloride Potent, selective mGlu5 antagonist MTEP hydrochloride
  74. BCC1795 Nepicastat Inhibitor of dopamine-β-hydroxylase,potent and selective Nepicastat
  75. BCC1808 NPS-2143 hydrochloride Selective antagonist of the calcium-sensing receptor; orally active calcilytic agent NPS-2143 hydrochloride
  76. BCC1819 Olmesartan Olmesartan
  77. BCC1822 ONO-AE3-208 High affinity and selective EP4 antagonist ONO-AE3-208
  78. BCC1823 Orteronel For castration-resistant prostate cancer, clinical candidate Orteronel
  79. BCC1828 Otenabant CB1 receptor antagonist Otenabant
  80. BCC1840 PB-22 Synthetic cannabinoid PB-22
  81. BCC1841 PD 123319 ditrifluoroacetate Angiotensin AT2 receptor antagonist PD 123319 ditrifluoroacetate
  82. BCC1845 Pentostatin Adenosine deaminase inhibitor Pentostatin
  83. BCC1854 PF-543 SphK1 inhibitor,cell-permeate,potent and selective PF-543
  84. BCC1868 Preladenant Adenosine A2A receptor antagonist Preladenant
  85. BCC1885 Reparixin Inhibitor of CXCL8 receptor and CXCR1/CXCR2 activation Reparixin
  86. BCC1886 Reparixin L-lysine salt CXCR1/CXCR2 inhibitor Reparixin L-lysine salt
  87. BCC1898 Rimonabant hydrochloride Selective CB1 receptor antagonist Rimonabant hydrochloride
  88. BCC1910 RS 504393 Highly selective CCR2 chemokine receptor antagonist RS 504393
  89. BCC1919 Salmefamol Salmefamol
  90. BCC1920 Salmeterol xinafoate β2-adrenergic receptor agonist Salmeterol xinafoate
  91. BCC1926 SB-222200 Potent, selective non-peptide NK3 antagonist. Brain penetrant SB-222200
  92. BCC1929 SB-408124 Hydrochloride OX1 receptor antagonist,selective and non-peptide SB-408124 Hydrochloride
  93. BCC1931 SB-674042 OX1 selective antagonist SB-674042
  94. BCC1932 SCH 527123 CXCR1 and CXCR2 receptors antagonist SCH 527123
  95. BCC1933 SCH 563705 CXCR2/CXCR1 antagonist,potent SCH 563705
  96. BCC1945 Setiptiline Serotonin receptor antagonist Setiptiline
  97. BCC1946 Setiptiline maleate Serotonin receptor antagonist Setiptiline maleate
  98. BCC1951 sitaxsentan Endothelin A (ETA) receptor antagonist sitaxsentan
  99. BCC1965 SRT3109 SRT3109
  100. BCC1966 SRT3190 CXCR2 ligand,SIRT1 activator SRT3190
  101. BCC1979 TAK-700 salt Androgen synthesis inhibitor TAK-700 salt

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