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Muscarinic Receptor

Muscarinic receptor is a group of G-protein coupled receptors that binds to acetylcholine and mediates cellular responses, including inhibition of acetylate cyclase, phosphoinositide degradation and regulation of potassium channels. It is involved in the neurological diseases such as Alzheimer's and Parkinson's.

Products for Muscarinic Receptor

  1. Cat.No. Product Name Information
  2. BCC1470 CevimelineMuscarinic receptor agonist
  3. BCC1471 Cevimeline hydrochloride hemihydrateAgonist of muscarinic receptor (M1/M3)
  4. BCC1516 DarifenacinM3 receptor antagonist and antimuscarinic agents
  5. BCC2022 Umeclidinium bromideMAChR antagonist
  6. BCC4565 Biperiden HClMuscarinic receptor antagonist; some selectivity for M1
  7. BCC4567 Darifenacin HBr
  8. BCC4575 Aclidinium BromideLAMAs antagonist
  9. BCC4580 Solifenacin succinateMuscarinic receptor antagonist
  10. BCC4583 5-hydroxymethyl Tolterodine (PNU 200577, 5-HMT, 5-HM)
  11. BCC4584 Fesoterodine Fumarate
  12. BCC4586 Tolterodine tartratePotent, non-selective muscarinic receptor antagonist
  13. BCC6164 VU 0365114Positive allosteric modulator of M5 receptors
  14. BCC6217 PTAC oxalateMuscarinic receptor ligand; exhibits partial agonist and antagonist activity at different subtypes
  15. BCC6627 Arecaidine but-2-ynyl ester tosylate
  16. BCC6628 Arecaidine propargyl ester tosylateMuscarinic agonist
  17. BCC6655 Nitrocaramiphen hydrochlorideMuscarinic antagonist, M1 > M2
  18. BCC6661 4-DAMPMuscarinic M3 antagonist
  19. BCC6682 W-84 dibromideStabilizer of cholinergic antagonist-receptor complexes
  20. BCC6707 5-MethylfurmethiodidePotent muscarinic agonist
  21. BCC6814 Oxotremorine sesquifumarateMuscarinic agonist
  22. BCC6920 Oxotremorine MMuscarinic agonist
  23. BCC6923 Pirenzepine dihydrochlorideSelective M1 muscarinic antagonist
  24. BCC6939 AF-DX 116Selective M2 antagonist
  25. BCC6946 Telenzepine dihydrochloridePotent, selective M1 antagonist
  26. BCC7024 AF-DX 384Potent M2/M4 antagonist
  27. BCC7042 McN-A 343Selective M1 muscarinic agonist
  28. BCC7061 (S)-(+)-Dimethindene maleateH1 antagonist. Also M2 muscarinic antagonist
  29. BCC7145 PD 102807Selective M4 antagonist
  30. BCC7263 DAU 5884 hydrochlorideM3 receptor antagonist
  31. BCC7314 AQ-RA 741Selective, high affinity M2 antagonist
  32. BCC7389 J 104129 fumaratePotent, selective M3 antagonist
  33. BCC7418 Zamifenacin fumarateSelective M3 antagonist
  34. BCC7427 Milameline hydrochlorideMuscarinic receptor agonist
  35. BCC7556 (+)-Muscarine iodideMuscarinic receptor agonist
  36. BCC7577 VU 10010
  37. BCC7729 VU 0238429Selective positive allosteric modulator of M5 receptors
  38. BCC7766 VU 0255035Highly selective muscarinic M1 antagonist
  39. BCC7907 VU 0357017 hydrochloridePositive allosteric modulator of M1 receptors

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