Home >> Research Area >> GPCR/G protein >> 5-HT Receptor

5-HT Receptor

5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.

Products for 5-HT Receptor

  1. Cat.No. Product Name Information
  2. BCC5224 Dihydroergotamine mesylate5-HT antagonist. Also partial agonist at adrenergic and dopaminergic D2 receptors
  3. BCC5247 Sarpogrelate hydrochlorideSelective 5-HT2A antagonist
  4. BCC5272 Ramosetron Hydrochloride
  5. BCC5421 Eltoprazine
  6. BCC5422 Eltoprazine hydrochloride5-HT2C receptor partial agonist
  7. BCC5423 RU 24969
  8. BCC5663 2-Methyl-5-hydroxytryptamine hydrochloride5-HT3 agonist/potent 5-HT6 ligand
  9. BCC5673 SB 203186 hydrochloride5-HT4 antagonist
  10. BCC5679 GR 466115-HT1D agonist
  11. BCC5680 m-CPP hydrochloride5-HT2B/2C receptor agonist
  12. BCC5693 RS 67333 hydrochloride5-HT4 partial agonist
  13. BCC5694 RS 39604 hydrochloride5-HT4 antagonist
  14. BCC5698 Methysergide maleate5-HT1/5-HT2 antagonist
  15. BCC5751 SB 200646 hydrochloride5-HT2C/2B antagonist
  16. BCC5752 SB 204070Potent and selective 5-HT4 antagonist
  17. BCC5925 DOI hydrochlorideMixed 5-HT2A/2C agonist
  18. BCC5937 SB 258719 hydrochlorideSelective 5-HT7 antagonist
  19. BCC5947 DOB hydrochlorideSelective 5-HT2 agonist
  20. BCC5949 SB 242084Selective 5-HT2C antagonist; brain penetrant
  21. BCC6035 SB 243213 dihydrochlorideSelective 5-HT2C inverse agonist
  22. BCC6127 MS 245 oxalateHigh affinity 5-HT6 antagonist
  23. BCC6168 PsilocinNon-selective serotonin receptor agonist
  24. BCC6194 AT 1015Long-acting 5-HT2A antagonist
  25. BCC6195 EMD 281014 hydrochlorideSelective 5-HT2A antagonist
  26. BCC6202 DV 7028 hydrochlorideSelective 5-HT2A antagonist; antithrombotic
  27. BCC6208 S 32212 hydrochloride
  28. BCC6265 PU 02Negative allosteric modulator of 5-HT3
  29. BCC6266 LP 20 hydrochlorideSelective 5-HT7 ligand
  30. BCC6291 Org 376845-HT2 agonist
  31. BCC6496 Cyclobenzaprine HCl5-HT2 receptor antagonist
  32. BCC6650 m-Chlorophenylbiguanide hydrochloridePotent and specific 5-HT3 agonist
  33. BCC6652 5-Carboxamidotryptamine maleateHas high affinity for 5-ht5A and 5-HT7. Also 5-HT1 agonist
  34. BCC6653 Cinanserin hydrochlorideSelective 5-HT2 antagonist
  35. BCC6678 4F 4PP oxalateSelective 5-HT2A antagonist
  36. BCC6691 Methylergometrine maleate
  37. BCC6696 α-Methyl-5-hydroxytryptamine maleate5-HT2B agonist
  38. BCC6697 N-Methylquipazine dimaleate5-HT3 agonist
  39. BCC6706 Methiothepin maleateHas moderate affinity for 5-ht5 and high affinity for 5-ht6 and 5-HT7. Also antagonist at 5-HT1 and 5-HT2
  40. BCC6709 MetergolineHas moderate affinity for 5-HT6 and high affinity for 5-HT7. Also 5-HT1/5-HT2 antagonist
  41. BCC6727 Quipazine dimaleate5-HT3 agonist
  42. BCC6733 MDL 722225-HT3 antagonist
  43. BCC6743 3-AQC5-HT3 antagonist
  44. BCC6767 RS 23597-190 hydrochloride5-HT4 antagonist
  45. BCC6771 2-[1-(4-Piperonyl)piperazinyl]benzothiazole5-HT4 agonist. Also 5-HT3 antagonist
  46. BCC6822 MDL 11,9395-HT2A antagonist
  47. BCC6856 MK 212 hydrochloride5-HT2C agonist
  48. BCC6870 1-Phenylbiguanide hydrochloride5-HT3 agonist
  49. BCC6877 RS 56812 hydrochloride5-HT3 partial agonist
  50. BCC6878 RS 67506 hydrochloride5-HT4 partial agonist
  51. BCC6882 Spiperone hydrochloride5-HT2A antagonist. Also D2-like antagonist
  52. BCC6887 N-Desmethylclozapine
  53. BCC6890 RS 16566 dihydrochloride5-HT3 ligand. Also shows affinity for zacopride binding site
  54. BCC6899 CP 93129 dihydrochloride5-HT1B agonist
  55. BCC6913 GR 55562 dihydrochloride5-HT1B antagonist
  56. BCC6915 BW 723C86 hydrochloride5-HT2B agonist
  57. BCC6967 SR 57227 hydrochloridePotent, selective 5-HT3 agonist
  58. BCC6976 SB 224289 hydrochlorideSelective 5-HT1B antagonist
  59. BCC6987 SB 216641 hydrochlorideSelective h5-HT1B antagonist
  60. BCC6994 SDZ SER 082 fumarateSelective 5-HT2B/2C antagonist
  61. BCC7018 CP 94253 hydrochloridePotent, selective 5-HT1B agonist
  62. BCC7019 GR 113808Potent, selective 5-HT4 antagonist
  63. BCC7035 SB 204741Potent, selective 5-HT2B antagonist
  64. BCC7036 SB 2283575-HT2C/2B antagonist/inverse agonist
  65. BCC7040 SB 221284Potent, selective 5-HT2C/2B antagonist
  66. BCC7056 NAS-181Selective r5-HT1B antagonist. Active in vivo
  67. BCC7081 GR 127935 hydrochloridePotent, selective 5-HT1B/1D antagonist
  68. BCC7101 LY 2158405-HT2/5-HT7 antagonist
  69. BCC7139 Mesulergine hydrochloride5-HT2A and 5-HT2C antagonist. Also dopamine receptor partial agonist
  70. BCC7142 GR 125487 sulfamatePotent, selective 5-HT4 antagonist; active in vivo
  71. BCC7143 SB 206553 hydrochloridePotent, selective 5-HT2C/5-HT2B antagonist. Orally active
  72. BCC7164 R-96544 hydrochloridePotent, selective 5-HT2A antagonist
  73. BCC7178 Zacopride hydrochloride5-HT4 agonist. Also highly potent 5-HT3 antagonist
  74. BCC7179 WAY 161503 hydrochloridePotent, selective 5-HT2C agonist
  75. BCC7183 Altanserin hydrochloride5-HT2A receptor antagonist
  76. BCC7196 Ro 60-0175 fumaratePotent, selective 5-HT2C agonist
  77. BCC7214 RitanserinPotent 5-HT2 antagonist
  78. BCC7216 SB 258585 hydrochloridePotent, selective 5-HT6 antagonist
  79. BCC7218 AS 19Potent 5-HT7 agonist
  80. BCC7222 PNU 142633Highly selective 5-HT1D agonist
  81. BCC7246 SDZ 205-557 hydrochloride5-HT4/5-HT3 receptor antagonist
  82. BCC7271 WAY 629 hydrochlorideSelective 5-HT2C agonist
  83. BCC7285 PNU 22394 hydrochloride5-HT2C agonist and 5-HT2A/2B partial agonist
  84. BCC7342 EMD 386088 hydrochloridePotent 5-HT6 agonist
  85. BCC7385 Melperone hydrochloride5-HT2A/D2 receptor antagonist; neuroleptic
  86. BCC7399 LP 44High affinity 5-HT7 agonist
  87. BCC7408 PNU 109291Potent and selective 5-HT1D agonist
  88. BCC7421 TCB-2Potent, high affinity 5-HT2A agonist
  89. BCC7437 L-703,664 succinateSelective 5-HT1D receptor agonist
  90. BCC7440 Fananserin5-HT2A antagonist. Also D4 antagonist
  91. BCC7479 Nefazodone hydrochloride5-HT uptake inhibitor and 5-HT2A antagonist. Antidepressant
  92. BCC7512 Ro 04-6790Potent and selective 5-HT6 antagonist
  93. BCC7517 LP 12 hydrochloride5-HT7 agonist
  94. BCC7536 1-MethylpsilocinPotent and selective 5-HT2C agonist
  95. BCC7558 LY 272015 hydrochlorideHigh affinity 5-HT2B antagonist; orally active
  96. BCC7559 LY 334370 hydrochlorideSelective 5-HT1F agonist
  97. BCC7562 CJ 033466Selective 5-HT4 partial agonist
  98. BCC7594 SB 699551Selective 5-ht5a antagonist
  99. BCC7595 SB 399885 hydrochloride
  100. BCC7629 NPS ALX Compound 4a dihydrochloridePotent and selective 5-HT6 antagonist
  101. BCC7650 BGC 20-761High affinity 5-HT6 antagonist
  102. BCC7660 LY 393558Dual 5-HT re-uptake inhibitor and 5-HT1B/1D antagonist
  103. BCC7695 ML 10302 hydrochloridePotent and selective 5-HT4 partial agonist
  104. BCC7718 Org 12962 hydrochlorideSelective 5-HT2C agonist
  105. BCC7742 Donitriptan hydrochloride5-HT1B/1D agonist
  106. BCC7750 SGS 518 oxalateSelective 5-HT6 antagonist
  107. BCC7774 CP 135807Selective 5-HT1D agonist
  108. BCC7807 WAY 208466 dihydrochlorideSelective 5-HT6 agonist
  109. BCC7836 NPEC-caged-serotoninCaged serotonin
  110. BCC7838 Zotepine5-HT2A/D2 antagonist; atypical antipsychotic
  111. BCC7856 LY 266097 hydrochlorideSelective 5-HT2B receptor antagonist
  112. BCC7877 MDL 100907Potent and selective 5-HT2A antagonist
  113. BCC7888 EMDT oxalateSelective 5-HT6 agonist
  114. BCC7919 ST 1936 oxalateSelective, high affinity 5-HT6 agonist
  115. BCC7928 BIMU 8Potent 5-HT4 receptor full agonist
  116. BCC7955 Tegaserod maleate5-HT4 partial agonist
  117. BCC7990 DR 4485 hydrochlorideHigh affinity and selective 5-HT7 antagonist; orally bioavailable
  118. BCC8025 NBOH-2C-CN hydrochlorideHigh affinity, selective 5-HT2A agonist
  119. BCC8065 Pimavanserin

Items 1 to 118 of 118 total