Products with Inhibitors bioactivity
| Cat.No. | Product Name |
|---|---|
| BCN3295 | Caffeic anhydride |
| 1. Caffeic anhydride can inhibit lipoxygenase in a concentration-dependent manner, with Ki values ranging from 0.85-57.6 microM. | |
| BCN3308 | Leachianone G |
| 1. Leachianone G shows inhibitory activities against pancreatic lipase, it may be used as drug candidate to control obesity. 2. (+/-)Leachianone G 1b, bearing 8-prenyl and 2',4'-dihydoxyl groups, exhibits potent vasorelaxant and neuroprotective effects. 3. Leachianone G exhibits significant antioxidant potentials in the ABTS, ONOO(-), and total ROS assays. 4. Leachianone G shows potent antiviral activity (IC(50) = 1.6 microg/ml). | |
| BCN3326 | 5-Methoxycanthin-6-one |
| 1. 5-Methoxycanthin-6-one exhibits a clear suppressive effect on the phagocytosis response upon activation with serum-opsonized zymosan in the range of IC₅₀ = 0.9-2.0 uM versus ibuprofen with IC₅₀ = 12.1 uM. 2. 5-Methoxycanthin-6-one displays moderate cytotoxic activity against the human prostate cancer cell PC-3 line, with IC₅₀ values ranging from 13.5-15.4 uM versus doxorubicine with IC₅₀ = 1.5 uM. | |
| BCN3334 | 6-Hydroxykaempferol |
| 1. 6-Hydroxykaempferol is a competitive inhibitor of tyrosinase compared to L-DOPA, it shows also high antioxidant activities. | |
| BCN3350 | Kushenol X |
| 1. Kushenol X exhibits inhibitory activity against Sodium-dependent glucose cotransporter 2(SGLT2). | |
