Products with Inhibitors bioactivity
| Cat.No. | Product Name |
|---|---|
| BCN3691 | Dihydroevocarpine |
| 1. Dihydroevocarpine and 1-methyl-2-undecyl-4-quinolone are moderate modulators of p-glycoprotein (p-gp) activity. 2. Dihydroevocarpine shows more potent inhibitory effects against MAO-B compared to MAO-A. 3. Dihydroevocarpine shows potent anti-Helicobacter pylori activity with the minimum inhibitory concentration (MIC) value of 10-20 microg/ml. | |
| BCN3693 | Mulberrofuran G |
| 1. Mulberrofuran G shows moderate activity, inhibits hepatitis B virus (HBV) DNA replication with the IC(50) value of 3.99 μM. | |
| BCN3697 | Benzyl 2,6-dimethoxybenzoate |
| 1. Benzyl 2,6-dimethoxybenzoate shows significant analgesic effects. 2. Benzyl 2,6-dimethoxybenzoate induces a concentration-dependent inhibition of the spontaneous contractions of the guinea-pig ileum with IC50 values ranging from 1.49 to 4.96 microM. 3. Benzyl 2,6-dimethoxybenzoate shows antimicrobial activity against several bacteria (S. aureus, E. coli, P. aeruginosa, and B. subtilis) and fungi (C. albicans and T. mentagrophytes). | |
| BCN3698 | Isoderrone |
| 1. Isoderrone is a protein tyrosine phosphatase 1B (PTP1B) inhibitor, with IC50 value of 22.7 ± 1.7 uM, suggests that it may be a new drug for treatment of type 2 diabetes. 2. Isoderrone shows inhibitory effects on α-glucosidase in vitro. | |
| BCN3702 | Panaxydiol |
| 1. Panaxydiol can inhibit rat liver cholesterol acyltransferase (ACAT) with IC50 values of 45 microM. | |
