Products with Inhibitors bioactivity
| Cat.No. | Product Name |
|---|---|
| BCN4857 | Atalantoflavone |
| 1. Atalantoflavone shows urease inhibitory potential. 2. Atalantoflavone displays weak cytotoxic activity against the human Caucasian prostate adenocarcinoma cell line PC-3. | |
| BCN4861 | 11-Hydroxytephrosin |
| 1. 11-Hydroxytephrosin inhibits NF-kappaB activity. | |
| BCN4866 | Pseudopalmatine |
| 1. Pseudopalmatine exhibits antiplasmodial activity. 2. Pseudopalmatine shows anti-acetylcholinesterase (AChE) activity, with IC50 values of 1.8uM. | |
| BCN4872 | Bavachin |
| Bavachin is a phytoestrogen that activates the estrogen receptors ERα and ERβ with EC50s of 320 and 680 nM, respectively. It is a cholesterol acyltransferase inhibitor, may have therapeutic potential for type 2 diabetes by activating insulin signaling pathways. Bavachin can stimulate the genetic expression of VEGF in PB,and directly help the fracture healing, and potentially protect cartilage from inflammation-mediated damage in joints of osteoarthritis patients through decreasing IL-1β-induced activation of IKK-IκBα-NF-κB signaling pathway. Bavachin has suppressive effects against pigmentation by melanin in the skin. | |
| BCN4881 | Xanthotoxol |
| Xanthotoxol shows strong pharmacological activities as anti-inflammatory, antioxidant, cytotoxic, dose-graded sedative, 5-HT antagonistic, and neuroprotective effects.Xanthotoxol also has calcium antagonistic effects, it blocks not only the voltage dependent calcium channel, but also the receptor operated calcium channel in the isolated guinea pig atria. | |
