Others Products Targets
- Oxidative Phosphorylation (6)
- NHE (3)
- Monocarboxylate Transporter (3)
- Matrix Metalloprotease (16)
- LXR-like Receptor (6)
- Voltage-gated Sodium (NaV) Channel (30)
- Voltage-gated Potassium (KV) Channel (38)
- Voltage-gated Calcium Channel (CaV) (38)
- Cell Adhesion Molecule (21)
- TRPV (30)
- Lipoxygenase (8)
- Bradykinin Receptor (12)
- Others (16)
- Cyclooxygenase (24)
- Apelin Receptor (5)
- TRPP (3)
- TRPML (3)
- TRPC (4)
- TRPA1 (7)
- Glycine Receptor (6)
- Epithelial Sodium Channel (3)
- STIM-Orai Channel (4)
- Ryanodine Receptor (6)
- Angiotensin-Converting Enzyme (8)
- 5-HT3 Receptor (39)
- IP3 Receptor (2)
- TRPM (8)
- Acid-Sensing Ion Channel (3)
- Calcium-Activated Potassium (KCa) Channel (19)
- VIP Receptor (7)
- Inward Rectifier Potassium (Kir) Channel (21)
- Stearoyl-CoA 9-Desaturase (1)
- Vasopressin Receptor (6)
- NADPH Oxidase (2)
- Monoamine Oxidase (10)
- Heme Oxygenase (2)
- NO donors and precursors (9)
- nNOS (5)
- iNOS (11)
- eNOS (1)
- Sodium and Potassium ATPase (3)
- KCC2 (1)
- H+-ATPase (3)
- Urotensin-II Receptor (8)
- H+,K+-ATPase (4)
- Ionophore (6)
- Chloride Channel (17)
- ETB Receptor (6)
- ETA Receptor (5)
- Angiotensin AT2 Receptor (3)
- Angiotensin AT1 Receptor (9)
- M5 Receptor (2)
- M4 Receptor (3)
- M3 Receptor (4)
- Purinergic (P2Y) Receptor (31)
- M2 Receptor (5)
- M1 Receptor (8)
- NCX (5)
- Ca2+-ATPase (7)
- Purinergic (P2X) Receptor (32)
- NKCC (2)
- Adrenergic α2 Receptor (33)
- Adrenergic α1 Receptor (22)
- HCN Channel (4)
- Adrenergic β3 Receptor (12)
- Adrenergic β2 Receptor (6)
- Adrenergic β1 Receptor (7)
- Protease-Activated Receptor (23)
- Prostanoid Receptor (24)
- Platelet-Activating Factor (PAF) Receptor (5)
- Phosphodiesterase (34)
Products for Others - Page 68
- Cat.No. Product Name Information/Activity
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BCN1035
Tetrodotoxin
Tetrodotoxin is a highly selective <b>sodium channel</b> blocker, with <b>IC<sub>50</sub></b> of 33 nM for <b>Nav1.6</b>.
-
BCC2156
Valproic acid sodium salt (Sodium valproate)
Valproic acid sodium salt (Sodium Valproate) is an HDAC inhibitor, with IC50 in the range of 0.5 and 2 mM, also inhibits HDAC1 (IC50, 400 μM), and induces proteasomal degradation of HDAC2. Valproic acid sodium salt activates Notch1 signaling and inhibits proliferation in small cell lung cancer (SCLC) cells. Valproic acid sodium salt is used in the treatment of epilepsy, bipolar disorder and prevention of migraine headaches.
-
BCC1048
β-Pompilidotoxin
Slows neuronal Na<sup>+</sup> channel inactivation
-
BCC5078
Rufinamide
Rufinamide(E 2080; CGP 33101; RUF 331) is a new antiepileptic agent that differs structurally from other antiepileptic drugs and is approved as adjunctive therapy for Lennox-Gastaut syndrome (LGS).
-
BCC4074
Icilin
Icilin(AG 3-5) is a synthetic super-agonist of TRPM8 ion channel.
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BCC6323
Optovin
Optovin is a reversible photoactive TRPA1 activator; stimulates human TRPA1 channels in vitro and enables repeated photoactivation of motor behaviors in wild-type zebrafish (EC50 = 2 μM).
-
BCC7597
Polygodial
6754-20-7
-
BCC7967
A 967079
A-967079 is a selective TRPA1 receptor antagonist with IC50s of 67 nM and 289 nM at human and rat TRPA1 receptors, respectively, and has good penetration into the CNS.
-
BCC7634
AP 18
Reversible TRPA1 channel blocker
-
BCC4910
HC-030031
HC-030031 is a potent and selective TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2±0.2 and 5.3±0.2 μM, respectively.
