Products with Inhibitors bioactivity
| Cat.No. | Product Name |
|---|---|
| BCN1134 | Oleoside |
| 1. Oleacein is a strong Angiotensin Converting Enzyme (ACE)-inhibitor (IC50 = 26 uM). | |
| BCN1143 | 4,5-Dimethoxycanthin-6-one |
| 4,5-Dimethoxycanthin-6-one has antibacterial actiyity, it exhibits inhibition against Staphylococcus aureus and its drug-resistant strains. 4,5-Dimethoxycanthin-6-one has a strong inhibitory effect on cyclic adenosine monophosphate (cAMP) phosphodiesterase. It also shows cytotoxicity against the tumor cell lines, U937 and HepG2. | |
| BCN1148 | Dimeric coniferyl acetate |
| 1. Dimeric coniferyl acetate shows strong NO inhibition with IC50 values of 27.1 uM in lipopolysacchalide (LPS)-activated murine macrophage-like J774.1 cells. 2. Dimeric coniferyl acetate exhibits significant inhibitory effects on the nitric oxide production in lipopolysaccharide activated C57BL6/J mouse macrophages. | |
| BCN1150 | Taxinine B |
| 1. Taxinine and taxinine B can inhibit the drug transport by P-glycoprotein in multidrug-resistant cells. 2. Taxinine B shows stronger inhibitory effects than acetylsalicylic acid (ASA) on platelet aggregation induced by arachidonic acid (AA). | |
| BCN1151 | Mangostanol |
| 1. Mangostanol has anti-cancer activity, it shows significant activities against the CEM-SS cell line, with IC50 values of 9.6 microg/ml. 2. Mangostanol is an acetylcholinesterase (AChE) selective inhibitor. | |
