Others - BioCrick

Cat.No. Product Name Information/Activity

BCC7769 RN 1747 RN-1747 is a selective transient receptor potential cation channel subfamily V member 4 (TRPV4) agonist, with EC50 values are 0.77 μM, 4.0 μM and 4.1 μM for hTRPV4, mTRPV4 and rTRPV4 respectively. RN-1747 also antagonizes TRPM8, with an IC50 of 4 μM. RN 1747 chemical structure

BCC6140 A 784168 Potent and selective TRPV1 antagonist A 784168 chemical structure

BCC1052 AMG-517 AMG 517 is a potent and selective vanilloid receptor-1 (TRPV1) antagonist with an IC50 of 0.5 nM. AMG-517 chemical structure

BCC7329 AMG 9810 AMG9810 is a selective and competitive vanilloid receptor 1 (TRPV1) antagonist with IC50 values of 24.5 and 85.6 nM for human and rat TRPV1, repectively. AMG 9810 chemical structure

BCC7500 Arachidonyl serotonin 187947-37-1 Arachidonyl serotonin chemical structure

BCC7797 BCTC BCTC is a potent and specific inhibitor of transient receptor potential cation channel subfamily M member 8 (TRPM8) in prostate cancer (PCa) DU145 cells. BCTC chemical structure

BCC1451 Capsazepine Capsazepine is a synthetic analogue of the sensory neurone excitotoxin, and an antagonist of TRPV1 receptor with an IC50 of 562 nM. Capsazepine chemical structure

BCC8009 GSK 2193874 GSK2193874 is an orally active, potent, and selective TRPV4 antagonist with IC50s of 2 nM and 40 nM for rTRPV4 and hTRPV4. GSK 2193874 chemical structure

BCC7861 HC 067047 HC-067047 is a potent and selective TRPV4 antagonist and reversibly inhibits currents through the human, rat, and mouse TRPV4 orthologs with IC50 values of 48 nM, 133 nM, and 17 nM, respectively. HC 067047 chemical structure

BCC5860 6-Iodonordihydrocapsaicin Potent, competitive vanilloid receptor antagonist 6-Iodonordihydrocapsaicin chemical structure

Others Products Targets

Products for Others - Page 20