5-HT2C Receptor
Serotonin 5-HT2C receptors, previously known as 5-HT1C receptors, are located primarily in the choroid plexus, cortex, limbic system and basal ganglia. 5-HT2C receptors play a role in CSF volume regulation, thermoregulation, penile erection and anxiety.
Products for 5-HT2C Receptor - Page 2
- Cat.No. Product Name Information/Activity
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BCC7179
WAY 161503 hydrochloride
276695-22-8
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BCC7271
WAY 629 hydrochloride
57756-44-2
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BCC5037
Clozapine
Clozapine (HF 1854) is an antipsychotic used to treat schizophrenia. Clozapine is a potent antagonist of dopamine and a number of other receptors, with a Ki of 9.5 nM for M1 receptor. Clozapine is also a potent and selective agonist at the muscarinic M4 receptor (EC50=11 nM).
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BCC1487
Clozapine N-oxide (CNO)
Activator of muscarinic DREAADs,Clozapine N-oxide is a pharmacologically inert metabolite of Clozapine, which is a potent <b>5-HT1C</b> receptor antagonist.
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BCC7139
Mesulergine hydrochloride
72786-12-0
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BCC6208
S 32212 hydrochloride
847871-78-7
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BCC5751
SB 200646 hydrochloride
143797-62-0
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BCC7143
SB 206553 hydrochloride
1197334-04-5
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BCC7040
SB 221284
196965-14-7
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BCC7036
SB 228357
SB228357 is a selective, potent oral active 5-HT2C/2B receptor antagonist with pKi values of 6.9, 8.0 and 9.0 for 5-HT2A, 5-HT2B and 5-HT2C, respectively. SB228357 has antidepressant/anxiolytic effects.
