GABAB Receptor
GABAB receptors are metabotropic G-protein-coupled receptors responsible for mediating the inhibitory effects of GABA alongside ionotropic GABAA and GABAA-ρ receptors. They exist as heterodimers of GABAB1 and GABAB2 subunits, with both required for function.
Products for GABAB Receptor - Page 2
- Cat.No. Product Name Information/Activity
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BCC5737
CGP 55845 hydrochloride
Potent, selective GABA<sub>B</sub> antagonist
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BCC6579
2-Hydroxysaclofen
117354-64-0
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BCC6562
Phaclofen
114012-12-3
-
BCC6580
Saclofen
125464-42-8
-
BCC5692
SCH 50911
SCH 50911, (+)-(S)-5,5-dimethylmorpholinyl-2-acetic acid, a selective, orally-active and competitive γ-Aminobutyric acid B GABA(B) receptor antagonist, binds to GABA(B) receptor with IC50 of 1.1 μM. SCH 50911 antagonizes GABA(B) autoreceptors, increasing the electrically-stimulated 3H overflow with an IC50 of 3 μM.
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BCC7644
rac BHFF
123557-91-5
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BCC7097
CGP 13501
Positive modulator at GABA<sub>B</sub> receptors
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BCC7096
CGP 7930
57717-80-3
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BCC7233
GS 39783
39069-52-8
-
BCC7186
N-ArachidonylGABA
128201-89-8
