GPBA Receptor
GPBA receptors (TGR5, GPBAR1, M-BAR) are G protein-coupled receptors (GPCRs) that are activated by bile acids. They are highly expressed in the gallbladder, ileum and colon, and are important in the regulation of glucose and lipid metabolism, and energy utilization.
Products for GPBA Receptor
- Cat.No. Product Name Information/Activity
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BCN5524
Betulinic acid
Betulinic acid is a natural pentacyclic triterpenoid, acts as a eukaryotic topoisomerase I inhibitor, with an IC50 of 5 μM, and possesses anti-HIV, anti-malarial, anti-inflammatory and anti-tumor properties. Betulinic acid acts as a new activator of NF-kB.
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BCC6201
GPBAR-A
GPBA receptor (TGR5) agonist
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BCN5616
Oleanolic acid
Oleanolic acid (Caryophyllin) is a natural compound from plants with anti-tumor activities.
