Search Site
Home >> Research Area >>GPCR/G protein>>Vasopressin Receptor >> (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

Catalog No. BCC6011
Size Price Stock
1mg $142.00 Ship Within 7 Days
Related Products

Organizitions Citing Our Products recently

 
 
 

Calcutta University

University of Minnesota

University of Maryland School of Medicine

University of Illinois at Chicago

The Ohio State University

University of Zurich

Harvard University

Colorado State University

Auburn University

Yale University

Worcester Polytechnic Institute

Washington State University

Stanford University

University of Leipzig

Universidade da Beira Interior

The Institute of Cancer Research

Heidelberg University

University of Amsterdam

University of Auckland
TsingHua University
TsingHua University
The University of Michigan
The University of Michigan
Miami University
Miami University
Jilin University
Jilin University
Fudan University
Fudan University
Wuhan University
Wuhan University
Sun Yat-sen University
Sun Yat-sen University
Universite de Paris
Universite de Paris

Quality Control of (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

Chemical structure

(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

Biological Activity of (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

Selective vasopressin V1A receptor antagonist. Inhibits vasopressin and oxytocin-induced increases in intracellular calcium concentrations in vitro (IC50 values are 5 and 30 nM respectively). Exhibits potent and prolonged antivasopressor activity and induces anxiolytic-like effects in the dorsal, but not ventral, hippocampus in vivo.

(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin Dilution Calculator

Concentration (start)
x
Volume (start)
=
Concentration (final)
x
Volume (final)
 
 
 
C1
V1
C2
V2

calculate

(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin Molarity Calculator

Mass
=
Concentration
x
Volume
x
MW*
 
 
 
g/mol

calculate

Chemical Properties of (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

Cas No. 73168-24-8 SDF Download SDF
Sequence YFQNCPRG

(Modifications: Tyr-1 = Pmp-Tyr(Me), Gly-8 = C-terminal amide)

Chemical Name (2S)-N-[(2S)-1-[(2-amino-2-oxoethyl)amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-1-[(10R,13S,16S,19S,22S)-13-(2-amino-2-oxoethyl)-16-(3-amino-3-oxopropyl)-19-benzyl-22-[(4-methoxyphenyl)methyl]-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentazaspiro[5.19]pentacosane-10-carbonyl]pyrrolidine-2-carboxamide
SMILES COC1=CC=C(C=C1)CC2C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(CSSC3(CCCCC3)CC(=O)N2)C(=O)N4CCCC4C(=O)NC(CCCN=C(N)N)C(=O)NCC(=O)N)CC(=O)N)CCC(=O)N)CC5=CC=CC=C5
Standard InChIKey QVQOGNOOAMQKCE-ZTYVOHGWSA-N
Standard InChI InChI=1S/C52H74N14O12S2/c1-78-32-16-14-31(15-17-32)25-35-46(73)63-36(24-30-10-4-2-5-11-30)47(74)61-34(18-19-40(53)67)45(72)64-37(26-41(54)68)48(75)65-38(29-79-80-52(27-43(70)60-35)20-6-3-7-21-52)50(77)66-23-9-13-39(66)49(76)62-33(12-8-22-58-51(56)57)44(71)59-28-42(55)69/h2,4-5,10-11,14-17,33-39H,3,6-9,12-13,18-29H2,1H3,(H2,53,67)(H2,54,68)(H2,55,69)(H,59,71)(H,60,70)(H,61,74)(H,62,76)(H,63,73)(H,64,72)(H,65,75)(H4,56,57,58)/t33-,34-,35-,36-,37-,38-,39-/m0/s1
Formula C52H74N14O12S2 M.Wt 1151.38
Solubility Soluble to 2 mg/ml in water
Storage Store at -20°C
General tips For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.
Shipping Condition Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.

Preparing Stock Solutions of (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

1 mg 5 mg 10 mg 20 mg 25 mg
1 mM 0.8685 mL 4.3426 mL 8.6852 mL 17.3705 mL 21.7131 mL
5 mM 0.1737 mL 0.8685 mL 1.737 mL 3.4741 mL 4.3426 mL
10 mM 0.0869 mL 0.4343 mL 0.8685 mL 1.737 mL 2.1713 mL
50 mM 0.0174 mL 0.0869 mL 0.1737 mL 0.3474 mL 0.4343 mL
100 mM 0.0087 mL 0.0434 mL 0.0869 mL 0.1737 mL 0.2171 mL
* Note: If you are in the process of experiment, it's necessary to make the dilution ratios of the samples. The dilution data above is only for reference. Normally, it's can get a better solubility within lower of Concentrations.

Kewords:

(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin,73168-24-8,GPCR/G protein,Vasopressin Receptor, supplier, inhibitor,Antagonist,Blocker,Modulator,Agonist, activators, activates, potent, BioCrick

Online Inquiry

Fill out the information below

* Required Fields

CheckCode: